Free Access
| Issue |
Med Sci (Paris)
Volume 28, Number 10, Octobre 2012
|
|
|---|---|---|
| Page(s) | 883 - 885 | |
| Section | Récepteurs couplés aux protéines G | |
| DOI | https://doi.org/10.1051/medsci/20122810018 | |
| Published online | 12 October 2012 | |
- Kenakin T. Agonist-receptor efficacy. II. Agonist trafficking of receptor signals. Trends Pharmacol Sci 1995 ; 16 : 232–238. [CrossRef] [PubMed] [Google Scholar]
- Allen JA, Yost JM, Setola V, et al. Discovery of beta-arrestin-biased dopamine D2 ligands for probing signal transduction pathways essential for antipsychotic efficacy. Proc Natl Acad Sci USA 2009 ; 108 : 18488–18493. [CrossRef] [Google Scholar]
- Galandrin S, Bouvier M. Distinct signaling profiles of beta1 and beta2 adrenergic receptor ligands toward adenylyl cyclase and mitogen-activated protein kinase reveals the pluridimensionality of efficacy. Mol Pharmacol 2006 ; 70 : 1575–1584. [CrossRef] [PubMed] [Google Scholar]
- Whalen EJ, Rajagopal S, Lefkowitz RJ. Therapeutic potential of beta-arrestin and G protein-biased agonists. Trends Mol Med 2011 ; 17 : 126–139. [CrossRef] [PubMed] [Google Scholar]
- Denis C, Saulière A, Galandrin S, et al. Probing heterotrimeric G protein activation: applications to biased ligands. Curr Pharm Des 2012 ; 18 : 128–144. [CrossRef] [PubMed] [Google Scholar]
- Verkaar F, van Rosmalen JW, Blomenröhr M, et al. G protein-independent cell-based assays for drug discovery on seven-transmembrane receptors. Biotechnol Annu Rev 2008 ; 14 : 253–274. [CrossRef] [PubMed] [Google Scholar]
- Saulière A, Bellot M, Paris H, et al. Deciphering biased-agonism complexity reveals a new active AT(1) receptor entity. Nat Chem Biol 2012 (sous presse). [Google Scholar]
- Wei H, Ahn S, Shenoy SK, et al. Independent beta-arrestin 2 and G protein-mediated pathways for angiotensin II activation of extracellular signal-regulated kinases 1 and 2. Proc Natl Acad Sci USA 2003 ; 100 : 10782–10787. [CrossRef] [Google Scholar]
Current usage metrics show cumulative count of Article Views (full-text article views including HTML views, PDF and ePub downloads, according to the available data) and Abstracts Views on Vision4Press platform.
Data correspond to usage on the plateform after 2015. The current usage metrics is available 48-96 hours after online publication and is updated daily on week days.
Initial download of the metrics may take a while.